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茆勇军 讲师
毕业单位 中科院上海药物研究所
办公电话 021-67791220
传真 021-67791214
联系地址 上海市龙腾路333号实训楼4413室
邮编 201620
电子邮箱 yongjun.mao@hotmail.com
所属团队 药物合成工艺团队
研究方向
主要从事药物合成工艺、药物发现领域的研究
个人经历
1997–2001, 沈阳药科大学,药物化学,学士;
2001–2004, 江苏扬子江药业市场部;
2004–2007, 沈阳药科大学,药物化学,硕士;
2007–2010, 中科院上海药物研究所,药物化学,博士;
2010–2012, State University of New York, Post Doctor of Medicinal Chemistry;
2012–, 上海工程技术大学化学化工学院,讲师
代表性论著(最新发表论文)
1. Yongjun Mao, Yang He, Fuqiang Zhu, Weiming Chen, Jingshan Shen, and Jianfeng Li*. New Synthesis of N-(4-Chloro-3-cyano-7-ethoxyquinolin-6-yl)acetamide. Heterocycles, 2014, 89(5), 1203–1209.
2. Yongjun Mao, Shuai Song, Dongmei Zhao,* and Maosheng Cheng. A New Total Synthesis of (±)-α-Noscapine. Heterocycles, 2013, 87(12), 2633–2640.
3. Yongjun Mao, Wenxiu Zhu, Xiaoguang Kong, Zhen Wang, Hua Xie, Jian Ding, Nicholas Kenneth Terrett, Jingkang Shen, Jingshan Shen. Design, synthesis and biological evaluation of novel pyrimidine, 3-cyanopyridine and m-amino-N-phenylbenzamide based monocyclic EGFR tyrosine kinase inhibitors. Bioorganic & Medicinal Chemistry, 2013, 12, 3090–3104.
4. Yongjun Mao, Nan Lin, Wang Tian, Ziwei Huang, and Jing An. New Synthesis of Pyrvinium that Inhibits the β-Catenin/Tcf4 Pathway. Heterocycles, 2012, 85(5), 1179–1185.
5. Yongjun Mao, Nan Lin, Wang Tian, Xiaofeng Han, Xiaobing Han, Ziwei Huang, and Jing An. Design, Synthesis and Biological Evaluation of New Diaminoquinazolines as β-Catenin/Tcf4 Pathway Inhibitors. Journal of Medicinal Chemistry, 2012, 55(3), 1346–1359.
6. Yongjun Mao, Zheng Liu, Xiaojun Yang, Xiangfei Xia, Rongxia Zhang, Jianfeng Li, Xiangrui Jiang, Kai Xie, Jin Zheng, Hui Zhang, Jin Suo, and Jingshan Shen. A New and Improved Process for N-(4-Chloro-3-cyano-7-ethoxyquinolin-6-yl)acetamide. Organic Process Research & Development, 2012, 16(12), 1970–1973.
科研成果
1.环丙胺类衍生物的不对称合成方法研究。上海高校青年教师培养资助计划(ZZGJD13017)。2014年1月-2015年12月。
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